Anastrozole (Arimidex)

Anastrozole is an anti estrogenic drug that is mostly being developed for the treatment of advanced breast cancer in women and is most commonly sold under trade name – Arimidex. Specifically, this agent is the first in a newer class of third generation selective oral aromatase inhibitors. Anastrozole is acting by blocking the enzyme aromatase, is subsequently blocking the production of the estrogen in the body.

Below you are going to find all the products containing Anastrozole and you’re also going to find a lot of information about this ingredient.

Show Filters

Showing all 13 results

Show Filters

Showing all 13 results

Due to the fact that many forms of breast cancer cells are being stimulated by the estrogen and its production, reducing the levels of this specific hormone in the body may greatly delay the progression of the disease. In addition to that, this is also be fundamental use of the tamoxifen citrate (for example Nolvadex), except for the fact that Nolvadex is blocking the action of estrogen at the receptor, not its actual endogenous production.

The effects of the Anastrozole (Arimidex) can be pretty much substantial, with a daily dosage of 1 mg (which is most often 1 tablet) that is capable of producing the estrogen suppression with more than 80% in most of the patients, therefore treating the issues.

With the very powerful effects that this product is having on the hormone levels in the human body, is very commonly only prescribed to post menopausal women since the effects it has are often believed to be “too powerful” in order to be prescribed to other people with other issues. Some side effects like for example hot flashes as well as hair thinning can present themselves during the therapy and it would be a lot much more worse and severe in the pre menopausal patients – one of the reasons why is often prescribed only to post menopausal women.

As in regards to the steroid-using male athlete (bodybuilder), anastrozole is a product that very often is being applied in order to minimize the side effects that are being associated with the elevated estrogen levels “thanks” to the anabolic/ androgenic steroid use that is often found as a big problem. Comparing it with the traditional methods like for example Nolvadex and Proviron, this product is a lot much more effective at controlling the estrogen levels in the body as is lowering the estrogen significantly better.

What Does Anastrozole Do?

What is Anastrozole? | What is Arimidex?

Anastrozole is an anti-estrogenic drug very often taken by bodybuilders in order to inhibit the estrogenic production. This agent is the first in a newer class of third generation selective oral aromatase inhibitors. Anastrozole is acting by blocking the enzyme aromatase, is subsequently blocking the production of the estrogen in the body.

What Are The Side Effects of Anastrozole?

The common side effects that can be associated with the use of an aromatase inhibitor (Anastrozole is in the AI family) is including: joint pain; mood changes; hot flashes; high blood pressure; weakness; headache; fatigue as well as swelling of the arms and/ or legs.

In addition to that, it was discovered that the AI’s are having some connection between the decreased bone mineral density therefore is believed they may decrease the bone mineral density. This effect may lead to a condition called osteoporosis and an increase in the factures in the susceptible patients. Some people out there also reported to have some gastrointestinal side effects in the time they are taking this medication so they are getting nausea and vomiting. It is very important to know that Aromatase Inhibitors can harm the development of an unborn fetus, therefore it never should be taken or handled during the pregnancy.

When Anastrozole is being taken by men (in the off label use) by trying to reduce the estrogen level in the time of the prolonged periods of the steroid treatment, the aromatase inhibitors (AI’s such as Anastrozole) may increase the cardiovascular disease (CVD) risk as well by taking away some of the good properties (benefits) of the hormone estrogen on the cholesterol values. It has been proven by different studies that when there’s an aromatizable steroid like for example testosterone enanthate that is being used along with an aromatase inhibitor, then the suppression of HDL (which is the good) cholesterol levels are becoming a lot much more noticed while the increase of LDL (bad) cholesterol gets more noticeable as well.

Due to the fact that the estrogen receptor agonist/ antagonist Nolvadex is generally not displaying the same anti estrogenic (negative) effect on the cholesterol values, it is normally favored over the aromatase inhibitors for the estrogen maintenance by the male bodybuilders and those athletes that are being concerned with the cardiovascular health.

Nonetheless, Anastrozole (Arimidex) is considered a much powerful anti estrogen product, therefore some people may favor Anastrozole over Novladex. It very much depends on everyone’s personal needs and health conditions.

How to Take Anastrozole?

Anastrozole (Arimidex) Administration

Anastrozole is a FDA approved drug for adjunctive treatment of postmenopausal women with hormone receptor- positive early breast cancer, first line treatment of postmenopausal women with hormone receptor- positive or receptor unknown locally advanced metastatic breast cancer as well as treatment of advanced breast cancer in postmenopausal women with disease progression following the tamoxifen therapy.

The dosage that is being prescribed in all of these examples is 1 mg per day and that’s until the progression of the disease is going to stop.

When it is being used in order to avoid the estrogenic side effects of the anabolic/ androgenic steroid use, the male athletes as well as bodybuilders are commonly using 0.5 mg to 1 mg of anastrozole per day as some people well respond to fight off with the side effects with only half a tablet while others need a full tablet. This mostly depends on the steroids used and on its dosages but also on how well a person responds to the drug either.

Anyway, in many cases only half of a tablet (which means 0.5 mg) taken every other day is quite enough to avoid the buildup of the estrogen. When is being used with readily aromatizing andogens like for example methandrostenolone or testosterone, such side effects as water retention (which can lead to high blood pressure) and gynecomastia are very often being blocked with great success. In addition to this, the use of the anastrozole may decrease the fat mass too, this can also be thanks to the connection with the estrogen levels.

The result can very often be a harder and much more defined appearance to the muscles as well as the physique, that is making that agent of an great interest for dieting and cutting reasons as well to a lot of bodybuilders out there. It should be taken in consideration the fact that food does not appear to affect the absorption of anastrozole, therefore the drug may be taken with or between meals as well.

Why Buy Anastrozole | Arimidex

Anastrozole (often sold as trade name - Arimidex) is an anti estrogenic drug that is very often used by male athletes in order to minimize the side effects that are being associated with the elevated estrogen levels that occur because of the anabolic/ androgenic steroid use. Anastrozole is a lot much more effective drug in controlling the estrogen level in comparison with the traditional methods.

Nonetheless, it has other side effects that are not associated with other anti estrogenic alternative drugs. For this reason, many people firstly try other alternative methods and in case they do not work, Anastrozole is among those drugs that are considered to work nearly for sure. For this reason, in case you are going to purchase Anastrozole, then there are nearly no chances that you are going to get wrong with it as it would work for sure.